Entry

Starting substrate

Product

Reflux Time (h)

Yield^a

(%)

1

3

quant

2

2

84

3

3

52

4

3

88

5

3

85

6

3

quant

7

3

94

8

2

quant

9

3

86

10

3

94

11

2

97

12

2.5

84